Weight management

Weight Loss Peptides

Weight loss peptides are not one bucket. Approved GLP-1 medicines, dual agonists, amylin analogs and investigational triple agonists sit at very different evidence levels.

Peptides covered
13
Highest evidence
5/5
Approved entries
7

How to compare this category

Use this page to compare the main weight loss peptides by mechanism, route, regulatory status and evidence quality before going deeper into the database entry or guide.

  • Prioritize approval status first: approved medications have regulated labels and larger safety datasets.
  • Treat investigational compounds as clinical-trial research, even when the early weight-loss numbers are strong.
  • Compare targets, not just pounds lost: GLP-1, GIP, glucagon and amylin pathways can produce different tolerability profiles.

Evidence scale

Scores rate evidence quality for the listed research context. They are not recommendations, prescriptions or a safety ranking.

Evidence 1/5
Mechanistic rationale only; no meaningful outcome evidence.
Evidence 2/5
Mostly animal, ex vivo, cell, or indirect evidence.
Evidence 3/5
Limited human pharmacology or small clinical evidence.
Evidence 4/5
Investigational compound with human randomized or phase 2/3 evidence.
Evidence 5/5
Approved medication with substantial human clinical evidence.
Weight Loss Peptides comparison table
PeptideStatusEvidenceBest forHalf-lifeActions
Retatrutide

Triple agonist (GLP-1 / GIP / glucagon)

Investigational
4/5

Phase 2 human evidence

Research comparison against GLP-1 and dual agonist drugs

Phase 2 human evidence; not approved

~6 days
Tirzepatide

Dual agonist (GLP-1 / GIP)

Approved
5/5

Approved with large human trials

Approved dual-incretin weight management reference

Approved medication with large clinical trials

~5 days
Semaglutide

GLP-1 receptor agonist

Approved
5/5

Approved with large human trials

Approved GLP-1 benchmark for weight loss and metabolic outcomes

Approved medication with large clinical trials

~7 days
Liraglutide

GLP-1 receptor agonist

Approved
5/5

Approved with human RCTs

Daily GLP-1 comparison and older approved option

Approved medication with human RCTs

~13 hours
Cagrilintide

Amylin analog

Investigational
4/5

Phase 2 human evidence

Amylin-pathway research and CagriSema context

Phase 2 human evidence; not approved

~7 days
Survodutide

Dual agonist (GLP-1 / glucagon)

Investigational
4/5

Human RCT evidence, investigational

GLP-1/glucagon research and MASH-adjacent context

Human RCT evidence; not approved

~7 days
HGH Fragment 176-191

Growth hormone C-terminal lipolytic fragment

Research only
2/5

Weak

General category comparison

See detail page for context.

Very short (minutes); poorly characterized
Dulaglutide

GLP-1 receptor agonist (Fc-fusion peptide)

Approved
5/5

Strong

General category comparison

See detail page for context.

Approximately 5 days
Exenatide

GLP-1 receptor agonist (incretin mimetic)

Approved
5/5

Approved drug, strong clinical evidence

General category comparison

See detail page for context.

Approximately 2.4 hours for immediate-release Byetta; extended-release (Bydureon BCise) microspheres release over weeks and exenatide can persist about 10 weeks after the last dose
Lixisenatide

Short-acting (prandial) GLP-1 receptor agonist; exendin-4-derived peptide

Approved
4/5

Approved drug with neutral cardiovascular outcomes; modest glycemic, not weight-loss, indication

General category comparison

See detail page for context.

Approximately 3 hours (reported range ~2.7-4.3 hours)
Albiglutide

GLP-1 receptor agonist (albumin-fusion)

Approved
4/5

Approved (later withdrawn); strong outcomes evidence

General category comparison

See detail page for context.

Approximately 5 days (reported terminal estimates ~5-8 days)
Efpeglenatide

GLP-1 receptor agonist (exendin-4-based)

Investigational
4/5

Strong trial evidence but investigational

General category comparison

See detail page for context.

Approximately 5.6 to 7.5 days (single-ascending-dose pharmacokinetic studies)
Adipotide

Pro-apoptotic peptidomimetic (vascular-targeting antiobesity agent)

Research only
2/5

Preclinical only; human program halted

General category comparison

See detail page for context.

Not well characterized in humans; dosed once daily by subcutaneous injection in animal and Phase 1 studies

Weight loss peptide cards

Retatrutide

Retatrutide

LY3437943

4/5

Research comparison against GLP-1 and dual agonist drugs

Phase 2 human evidence; not approved

Tirzepatide

Tirzepatide

LY3298176, Mounjaro, Zepbound

5/5

Approved dual-incretin weight management reference

Approved medication with large clinical trials

Semaglutide

Semaglutide

Ozempic, Wegovy, Rybelsus

5/5

Approved GLP-1 benchmark for weight loss and metabolic outcomes

Approved medication with large clinical trials

Liraglutide

Liraglutide

Victoza, Saxenda

5/5

Daily GLP-1 comparison and older approved option

Approved medication with human RCTs

Survodutide

Survodutide

BI 456906

4/5

GLP-1/glucagon research and MASH-adjacent context

Human RCT evidence; not approved

HGH Fragment 176-191

HGH Fragment 176-191

HGH Frag 176-191

2/5

A synthetic C-terminal fragment of human growth hormone claimed to stimulate adipocyte lipolysis without binding the GH receptor or raising IGF-1, though human fat-loss evidence is weak.

Growth hormone C-terminal lipolytic fragment

Dulaglutide

Dulaglutide

Trulicity

5/5

Dulaglutide is a long-acting GLP-1 receptor agonist that stimulates glucose-dependent insulin secretion, suppresses glucagon, slows gastric emptying and reduces appetite.

GLP-1 receptor agonist (Fc-fusion peptide)

Exenatide

Exenatide

Byetta, Bydureon, exendin-4

5/5

Exenatide activates the GLP-1 receptor to increase glucose-dependent insulin secretion, suppress inappropriate glucagon release, and slow gastric emptying.

GLP-1 receptor agonist (incretin mimetic)

Lixisenatide

Lixisenatide

Adlyxin, Lyxumia

4/5

Lixisenatide is an exendin-4-derived GLP-1 receptor agonist that slows gastric emptying and lowers postprandial glucose while stimulating glucose-dependent insulin release and suppressing glucagon.

Short-acting (prandial) GLP-1 receptor agonist; exendin-4-derived peptide

Albiglutide

Albiglutide

Tanzeum, Eperzan

4/5

Albiglutide is a long-acting GLP-1 receptor agonist made by fusing two DPP-4-resistant copies of modified human GLP-1 to recombinant human albumin, activating the GLP-1 receptor to boost glucose-dependent insulin secretion and suppress glucagon.

GLP-1 receptor agonist (albumin-fusion)

Efpeglenatide

Efpeglenatide

LY3434285

4/5

An exendin-4-based GLP-1 receptor agonist conjugated to an antibody Fc fragment that slows clearance and activates the GLP-1 receptor to boost glucose-dependent insulin secretion, slow gastric emptying and reduce appetite.

GLP-1 receptor agonist (exendin-4-based)

Adipotide

Adipotide

FTPP, prohibitin-targeting peptide

2/5

Adipotide is a chimeric peptidomimetic whose CKGGRAKDC homing motif binds prohibitin on white-fat blood-vessel endothelium, where its fused D(KLAKLAK)2 segment disrupts mitochondrial membranes to trigger endothelial apoptosis and regression of the fat tissue's blood supply.

Pro-apoptotic peptidomimetic (vascular-targeting antiobesity agent)

Weight loss guides

Read the strongest related guides for this category before drilling into a single database entry.

FAQ

What are the best-studied weight loss peptides?

Semaglutide, liraglutide and tirzepatide have the strongest human evidence because they are approved medications with large randomized trials and regulated labels.

Are retatrutide and cagrilintide approved for weight loss?

No. Retatrutide and cagrilintide have human trial evidence, but they remain investigational and should be treated as research compounds until regulators approve a label.

How should weight loss peptides be compared?

Compare approval status, trial evidence, mechanism, adverse-effect profile, dosing schedule and contraindications. Weight-loss percentage alone is not enough context.

More peptide categories

Research & educational purposes only

The information on PeptideStat is for educational and research purposes only and is not medical advice. Many peptides discussed are research compounds not approved for human use. Always consult a qualified healthcare professional before making any health decisions. Articles may contain affiliate links — we may earn a commission at no extra cost to you.